Frank E. Kwarcinski
Biochemistry, Genetics and Molecular Biology · University of Michigan
Publications
46
Citations
517
Est. group size
~3
Recurring co-author estimate
Active years
16
Publishing since 2011
Typically publishes in teams of ~13 · 6% small-team papers (≤3 authors) · across 12 venues
- Identification of 4‐Anilinoquin(az)oline as a Cell‐Active Protein Kinase Novel 3 (PKN3) Inhibitor Chemotype
UNC Libraries · 2025
- Structures of Ric-8B in complex with Gα protein folding clients reveal isoform specificity mechanisms
Structure · 2023
- Characterization of 2,4-Dianilinopyrimidines Against Five <i>P. falciparum</i> Kinases PfARK1, PfARK3, PfNEK3, PfPK9, and PfPKB
ACS Medicinal Chemistry Letters · 2023
- SGC-CLK-1: A chemical probe for the Cdc2-like kinases CLK1, CLK2, and CLK4
Current Research in Chemical Biology · 2023
- Characterization of 2,4-dianilinopyrimidines Against Five P. falciparum Kinases PfARK1, PfARK3, PfNEK3, PfPK9 and PfPKB
ChemRxiv · 2023
- Discovery of potent Plasmodium falciparum protein kinase 6 (PfPK6) inhibitors with a type II inhibitor pharmacophore
European Journal of Medicinal Chemistry · 2022
- Identification of Novel 2,4,5-Trisubstituted Pyrimidines as Potent Dual Inhibitors of Plasmodial <i>Pf</i> GSK3/ <i>Pf</i> PK6 with Activity against Blood Stage Parasites In Vitro
Journal of Medicinal Chemistry · 2022
- Identification of 4‐Anilinoquin(az)oline as a Cell‐Active Protein Kinase Novel 3 (PKN3) Inhibitor Chemotype**
ChemMedChem · 2022
- Discovery of Potent Plasmodium falciparum Protein Kinase 6 (PfPK6) Inhibitors with a Type II Inhibitor Pharmacophore
ChemRxiv · 2022
- Structures of Ric-8B in Complex With Gα Protein Folding Clients Reveal Isoform Specificity Mechanisms
SSRN Electronic Journal · 2022
- Identification of Novel 2,4,5-Trisubstituted Pyrimidines as Potent Dual Inhibitors of Plasmodial PfGSK3/PfPK6 with Activity Against Blood Stage Parasites in vitro
ChemRxiv · 2022
- SGC-CLK-1 (CAF-170) a chemical probe for the Cdc2-Like kinases CLK1, CLK2, and CLK4
bioRxiv (Cold Spring Harbor Laboratory) · 2022
- A Chemical Probe for Dark Kinase STK17B Derives Its Potency and High Selectivity through a Unique P-Loop Conformation
Journal of Medicinal Chemistry · 2020
- Identification and Optimization of cell active 4-anilino-quin(az)oline Inhibitors for Protein Kinase Novel 3 (PKN3)
bioRxiv (Cold Spring Harbor Laboratory) · 2020
- A Chemical Probe for Dark Kinase STK17B Derives its Potency and High Selectivity Through a Unique P-loop Conformation
ChemRxiv · 2020
- ChemRxiv×5
- bioRxiv (Cold Spring Harbor Laboratory)×4
- ACS Chemical Biology×2
- Journal of Medicinal Chemistry×2
- Clinical Cancer Research×2
- Matthew Clark
Biochemistry, Genetics and Molecular Biology · Purdue University West Lafayette
- Stuart J. Decker
Biochemistry, Genetics and Molecular Biology · University of Michigan
- Alan V. Smrcka
Biochemistry, Genetics and Molecular Biology · University of Michigan
- Angeline M. Lyon
Biochemistry, Genetics and Molecular Biology · Purdue University West Lafayette
- Behirda Karaj
Biochemistry, Genetics and Molecular Biology · University of Michigan
This profile was generated automatically from public scholarly data (OpenAlex). Group size and activity levels are estimates derived from co-authorship patterns.
Last updated Jul 25, 2026.
Claim or correct this profile